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Le mГ©canisme d'action prГ©cis n'est pas complГЁtement compris, mais le modafinil agit comme un inhibiteur de la recapture de la sГ©rotonine et un agoniste partiel des rГ©cepteurs de la sГ©rotonine. Il agit dans le cortex cГ©rГ©bral, l'hypothalamus et le tegmentum du cerveau. C'est un stimulant doux avec un dГ©but d'action trГЁs rapide. Tous les animaux (rats et souris) de l'Г©tude ont dormi davantage aprГЁs avoir pris du Modafinil. Un autre modafinil commercialisГ©, que la sociГ©tГ© vend sous le nom de В« Provigil Professional 200 В», est destinГ© aux travailleurs postГ©s.
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Les effets secondaires rares et graves peuvent inclure l'anaphylaxie et le syndrome de Stevens-Johnson, ainsi que des hallucinations chez les personnes ayant des antГ©cГ©dents de psychose. Il n'est pas clair si l'utilisation pendant la grossesse est sans danger. Les stimulants peuvent augmenter la frГ©quence cardiaque et la pression artГ©rielle et les patients qui utilisent Modafinil peuvent signaler une augmentation de la frГ©quence cardiaque. On pense que cet agent agit en modulant directement ou indirectement la voie de l'adГ©nosine.
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